99% Tianeptine sodium masima CAS 30123-17-2
Fa'amatalaga
MEA | TULAGA | i'uga |
Fa'aaliga | Pa'epa'e i le pa'epa'e samasama | Pa'epa'e tioata pa'epa'e |
Solubility | Solufua saoloto I le vai ma methanol ma le dichloromethane | Fa'atatau |
Fa'ailoaga | E IR, Ina ia fetaui ma tulaga faigaluega | Fa'atatau |
(2) E maua ai le tali ole sodium | Fa'atatau | |
Fa'aleaga A | ≤0.1% | Le iloa |
Fa'atasiga fa'atasi | So'o se Max tasi le mama≤0.1% | 0.060% |
Aofa'iga o mea leaga≤0.4% | 0.36% | |
Solvents totoe (GC) | Acetidin≤ 0.5% | ND |
Dichloromethane≤ 0.06% | ND | |
Methanol≤ 0.3% | ND | |
Acetone≤ 0.5% | 0.29% | |
Acetonitrile≤0.041% | 0.022% | |
Ethanol≤0.5% | ND | |
N, N-dimethylformamide≤0.088% | ND | |
Vai | ≤ 5.0% | 3.8% |
Su'ega (HPLC) | 99.0%-101.0% (I luga o le anhydrousbasis) | 99.70% |
Fa'aaogāga
Tianeptine sodiummasimaose tricyclic antidepressant.O lona faiga fa'ama'i e 'ese'ese mai le fa'ama'i fa'ama'i fa'amasani tricyclic.E mafai ona faʻateleina le toe faʻaleleia o le 5-HT i le synaptic cleft.Aafiaga ole HT neuronal conduction.Leai se sootaga mo choline poʻo adrenergic receptors.Ole malosi ole antidepressant e tutusa ma le tricyclics, ae o le tolerability e sili atu nai lo tricyclics.Mo le togafitiga o le vaivai, feololo poʻo le ogaoga o le atuatuvale, neurogenic ma le faʻalavelave faʻalavelave, popole ma le atuatuvale faʻatasi ma le tino, aemaise lava le faʻafitauli o le manava, ma le popole ma le atuatuvale i tagata mamaʻi faʻalagolago i le ava i le taimi o le toesea.